Lead optimization

Lead optimization is an operationally diverse stage of the drug discovery process in which the chemical structures of compounds or biologics are modified to improve target specificity and selectivity, plus pharmacodynamic, pharmacokinetic, and toxicological properties to produce a preclinical drug candidate. This process requires detailed characterization of lead compound series and lead biologics, including data related to toxicity, efficacy, stability, and bioavailability.

  • Biotherapeutics
  • Cheminformatics
  • Fragment-based lead discovery

Related Conference of Lead optimization

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14th International Conference on Chemistry Meeting

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